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Optimization of the aminopyridopyrazinones class of PDE5 inhibitors: Discovery of 3-[(trans-4-hydroxycyclohexyl)amino]-7-(6-methoxypyridin-3-yl)-1-(2-propoxyethyl)pyrido[3,4-b]pyrazin-2(1H)-one
Robert O. Hughes, John K. Walker, D. Joseph Rogier, Steve E. Heasley, Rhadika M. Blevis-Bal, Alan G. Benson, E. Jon Jacobsen, Jerry W. Cubbage, Yvette M. Fobian, Dafydd R. Owen, John N. Freskos, JohnVolume:
19
Year:
2009
Language:
english
Pages:
5
DOI:
10.1016/j.bmcl.2009.07.019
File:
PDF, 816 KB
english, 2009