Replacement of pyrazol-3-yl amine hinge binder with thiazol-2-yl amine: Discovery of potent and selective JAK2 inhibitors
Stephanos Ioannidis, Michelle L. Lamb, Lynsie Almeida, Huiping Guan, Bo Peng, Geraldine Bebernitz, Kirsten Bell, Marat Alimzhanov, Michael ZindaVolume:
20
Year:
2010
Language:
english
Pages:
5
DOI:
10.1016/j.bmcl.2010.01.091
File:
PDF, 459 KB
english, 2010