Intrinsic electrophilicity of the 4-methylsulfonyl-2-pyridone scaffold in glucokinase activators: Role of glutathione-S-transferases and in vivo quantitation of a glutathione conjugate in rats
John Litchfield, Raman Sharma, Karen Atkinson, Kevin J. Filipski, Stephen W. Wright, Jeffrey A. Pfefferkorn, Beijing Tan, Rachel E. Kosa, Benjamin Stevens, Meihua Tu, Amit S. KalgutkarVolume:
20
Year:
2010
Language:
english
Pages:
6
DOI:
10.1016/j.bmcl.2010.08.095
File:
PDF, 689 KB
english, 2010