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Imidazo[4,5-d]thiazolo[5,4-b]pyridine based inhibitors of IKK2: Synthesis, SAR, PK/PD and activity in a preclinical model of rheumatoid arthritis
Alaric J. Dyckman, Charles M. Langevine, Claude Quesnelle, James Kempson, Junqing Guo, Patrice Gill, Steven H. Spergel, Scott H. Watterson, Tianle Li, David S. Nirschl, Kathleen M. Gillooly, Mark A. PVolume:
21
Year:
2011
Language:
english
Pages:
4
DOI:
10.1016/j.bmcl.2010.10.133
File:
PDF, 1.56 MB
english, 2011