Fragmentation of GW4064 led to a highly potent partial farnesoid X receptor agonist with improved drug-like properties
Flesch, Daniel, Gabler, Matthias, Lill, Andreas, Gomez, Roberto Carrasco, Steri, Ramona, Schneider, Gisbert, Stark, Holger, Schubert-Zsilavecz, Manfred, Merk, DanielVolume:
23
Language:
english
Journal:
Bioorganic & Medicinal Chemistry
DOI:
10.1016/j.bmc.2015.04.035
Date:
July, 2015
File:
PDF, 798 KB
english, 2015