3,4-Diaza-bicyclo[4.1.0]hept-4-en-2-one phenoxypropylamine analogs of irdabisant (CEP-26401) as potent histamine-3 receptor inverse agonists with robust wake-promoting activity
Hudkins, Robert L., Becknell, Nadine C., Lyons, Jacquelyn A., Aimone, Lisa D., Olsen, Mark, Haltiwanger, R. Curtis, Mathiasen, Joanne R., Raddatz, Rita, Gruner, John A.Volume:
95
Language:
english
Journal:
European Journal of Medicinal Chemistry
DOI:
10.1016/j.ejmech.2015.03.054
Date:
May, 2015
File:
PDF, 639 KB
english, 2015