Discovery of (1 R ,2 S )-2-{[(2,4-Dimethylpyrimidin-5-yl)oxy]methyl}-2-(3-fluorophenyl)- N -(5-fluoropyridin-2-yl)cyclopropanecarboxamide (E2006): A Potent and Efficacious Oral Orexin Receptor Antagonist
Yoshida, Yu, Naoe, Yoshimitsu, Terauchi, Taro, Ozaki, Fumihiro, Doko, Takashi, Takemura, Ayumi, Tanaka, Toshiaki, Sorimachi, Keiichi, Beuckmann, Carsten T., Suzuki, Michiyuki, Ueno, Takashi, Ozaki, ShVolume:
58
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.5b00217
Date:
June, 2015
File:
PDF, 2.88 MB
english, 2015