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Optimization of a novel series of N-phenylindoline-5-sulfonamide-based acyl CoA:monoacylglycerol acyltransferase-2 inhibitors: Mitigation of CYP3A4 time-dependent inhibition and phototoxic liabilities
Sato, Kenjiro, Takahagi, Hiroki, Kubo, Osamu, Hidaka, Kousuke, Yoshikawa, Takeshi, Kamaura, Masahiro, Nakakariya, Masanori, Amano, Nobuyuki, Adachi, Ryutaro, Maki, Toshiyuki, Take, Kazumi, Takekawa, SVolume:
23
Language:
english
Journal:
Bioorganic & Medicinal Chemistry
DOI:
10.1016/j.bmc.2015.06.003
Date:
August, 2015
File:
PDF, 925 KB
english, 2015