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Discovery of a novel tricyclic 4H-thiazolo[5′,4′:4,5]pyrano[2,3-c]pyridine-2-amino scaffold and its application in a PI3Kα inhibitor with high PI3K isoform selectivity and potent cellular activity
Gerspacher, Marc, Fairhurst, Robin A., Mah, Robert, Roehn-Carnemolla, Esther, Furet, Pascal, Fritsch, Christine, Guthy, Daniel A.Volume:
25
Language:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2015.06.077
Date:
September, 2015
File:
PDF, 530 KB
english, 2015