An optimized polyamine moiety boosts the potency of human type II topoisomerase poisons as quantified by comparative analysis centered on the clinical candidate F14512
Palermo, Giulia, Minniti, Elirosa, Greco, Maria Laura, Riccardi, Laura, Simoni, Elena, Convertino, Marino, Marchetti, Chiara, Rosini, Michela, Sissi, Claudia, Minarini, Anna, De Vivo, MarcoYear:
2015
Language:
english
Journal:
Chem. Commun.
DOI:
10.1039/C5CC05065K
File:
PDF, 2.14 MB
english, 2015