Synthesis, Biological Activity and Molecular Modeling Studies of 1,2,3,4-Tetrahydroiso-quinoline Derivatives as Conformationally Constrained Analogues of KN62, a Potent Antagonist of the P2X7-Receptor Containing a Tyrosine Moiety
Baraldi, Pier, Makaeva, Rimma, Pavani, Maria, Nuñez, Maria, Spalluto, Giampiero, Moro, Stefano, Falzoni, Simonetta, Virgilio, Francesco, Romagnoli, RomeoVolume:
52
Language:
english
Journal:
Arzneimittelforschung
DOI:
10.1055/s-0031-1299891
Date:
December, 2011
File:
PDF, 252 KB
english, 2011