Brain accumulation of the EML4-ALK inhibitor ceritinib is restricted by P-glycoprotein (P-GP/ABCB1) and breast cancer resistance protein (BCRP/ABCG2)
Kort, Anita, Sparidans, Rolf W., Wagenaar, Els, Beijnen, Jos H., Schinkel, Alfred H.Language:
english
Journal:
Pharmacological Research
DOI:
10.1016/j.phrs.2015.09.003
Date:
September, 2015
File:
PDF, 785 KB
english, 2015