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Comprehensive Analysis of Structure–Activity Relationships of α-Ketoheterocycles as sn -1-Diacylglycerol Lipase α Inhibitors
Janssen, Freek J., Baggelaar, Marc P., Hummel, Jessica J. A., Overkleeft, Herman S., Cravatt, Benjamin F., Boger, Dale L., van der Stelt, MarioLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.5b01627
Date:
December, 2015
File:
PDF, 1.12 MB
english, 2015