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Discovery of potent aryl-substituted 3-[(3-methylpyridine-2-carbonyl) amino]-2,4-dimethyl-benzoic acid EP4 antagonists with improved pharmacokinetic profile
Blanco, Maria-Jesus, Vetman, Tatiana, Chandrasekhar, Srinivasan, Fisher, Matthew J., Harvey, Anita, Chambers, Mark, Lin, Chaohua, Mudra, Daniel, Oskins, Jennifer, Wang, Xu-Shan, Yu, Xiao-Peng, WarshawLanguage:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2015.12.057
Date:
December, 2015
File:
PDF, 405 KB
english, 2015