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A Poised Fragment Library Enables Rapid Synthetic Expansion Yielding the First Reported Inhibitors of PHIP(2), an Atypical Bromodomain
Cox, Oakley B, Krojer, Tobias, Collins, Patrick, Monteiro, Octovia, Talon, Romain, Bradley, Anthony, Fedorov, Oleg, Marsden, Brian, Amin, Jahangir, Spencer, John, von Delft, Frank, Brennan, PaulYear:
2015
Language:
english
Journal:
Chem. Sci.
DOI:
10.1039/C5SC03115J
File:
PDF, 1.86 MB
english, 2015