Discovery and preclinical evaluation of potent, orally bioavailable, metabolically stable cyclopropylindolobenzazepine acylsulfonamides as thumb site 1 inhibitors of the hepatitis c virus NS5B RNA-dependent, RNA polymerase
Hewawasam, Piyasena, Tu, Yong, Gao, Min, Hanumegowda, Umesh, Knipe, Jay, Lemm, Julie A., Parker, Dawn D., Rigat, Karen L., Roberts, Susan B., Meanwell, Nicholas A., Kadow, John F.Language:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2015.12.058
Date:
December, 2015
File:
PDF, 556 KB
english, 2015