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A phenotypic drug discovery study on thienodiazepine derivatives as inhibitors of T cell proliferation induced by CD28 co-stimulation leads to the discovery of a first bromodomain inhibitor
Endo, Junichi, Hikawa, Hidemasa, Hamada, Maiko, Ishibuchi, Seigo, Fujie, Naoto, Sugiyama, Naoki, Tanaka, Minoru, Kobayashi, Haruhito, Sugahara, Kunio, Oshita, Koichi, Iwata, Kazunori, Ooike, Shinsuke,Volume:
26
Language:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2016.01.084
Date:
March, 2016
File:
PDF, 1.27 MB
english, 2016