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Discovery of 5-Chloro-1-(5-chloro-2-(methylsulfonyl)benzyl)-2-imino-1,2-dihydropyridine-3-carboxamide (TAK-259), as a Novel, Selective, and Orally Active α1D Adrenoceptor Antagonist with Anti−urinary Frequency Effects: Reducing Human Ether−a−go−go−Related Gene (hERG) Liabilities
Sakauchi, Nobuki, Kohara, Yasuhisa, Sato, Ayumu, Suzaki, Tomohiko, Imai, Yumi, Okabe, Yuichi, Imai, Shigemitsu, Saikawa, Reiko, Nagabukuro, Hiroshi, Kuno, Haruhiko, Fujita, Hisashi, Kamo, Izumi, YoshiLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.5b01528
Date:
March, 2016
File:
PDF, 723 KB
english, 2016