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Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit
Gerstenberger, Brian S., Trzupek, John D., Tallant, Cynthia, Fedorov, Oleg, Filippakopoulos, Panagis, Brennan, Paul E., Fedele, Vita, Martin, Sarah, Picaud, Sarah, Rogers, Catherine, Parikh, Mihir, TaLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.6b00012
Date:
May, 2016
File:
PDF, 9.24 MB
english, 2016