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Telescoped Process to Manufacture 6,6,6-Trifluorofucose via Diastereoselective Transfer Hydrogenation: Scalable Access to an Inhibitor of Fucosylation Utilized in Monoclonal Antibody Production
Achmatowicz, Michal M., Allen, John G., Bio, Matthew M., Bartberger, Michael D., Borths, Christopher J., Colyer, John T., Crockett, Richard D., Hwang, Tsang-Lin, Koek, Jan. N., Osgood, Stephen A., RobLanguage:
english
Journal:
The Journal of Organic Chemistry
DOI:
10.1021/acs.joc.6b00646
Date:
May, 2016
File:
PDF, 980 KB
english, 2016