Structural modifications of the serotonin 5-HT7 receptor agonist N-(4-cyanophenylmethyl)-4-(2-biphenyl)-1-piperazinehexanamide (LP-211) to improve in vitro microsomal stability: A case study
Lacivita, Enza, Podlewska, Sabina, Speranza, Luisa, Niso, Mauro, Satała, Grzegorz, Perrone, Roberto, Perrone-Capano, Carla, Bojarski, Andrzej J., Leopoldo, MarcelloLanguage:
english
Journal:
European Journal of Medicinal Chemistry
DOI:
10.1016/j.ejmech.2016.05.005
Date:
May, 2016
File:
PDF, 1.51 MB
english, 2016