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Furoates and thenoates inhibit pyruvate dehydrogenase kinase 2 allosterically by binding to its pyruvate regulatory site
Masini, Tiziana, Birkaya, Barbara, van Dijk, Simon, Mondal, Milon, Hekelaar, Johan, Jäger, Manuel, Terwisscha van Scheltinga, Anke C., Patel, Mulchand S., Hirsch, Anna K. H., Moman, EdelmiroLanguage:
english
Journal:
Journal of Enzyme Inhibition and Medicinal Chemistry
DOI:
10.1080/14756366.2016.1201812
Date:
July, 2016
File:
PDF, 506 KB
english, 2016