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Discovery of N-((1-(4-(3-(3-((6,7-dimethoxyquinolin-3-yl)oxy)phenyl)ureido)-2-(trifluoromethyl)phenyl)piperidin-4-yl)methyl)propionamide (CHMFL-KIT-8140) as a Highly Potent Type II Inhibitor Capable of Inhibiting the T670I “Gatekeeper” Mutant of cKIT Kinase
Li, Binhua, Wang, Aoli, Liu, Juan, Qi, Ziping, Liu, Xiaochuan, Yu, Kailin, Wu, Hong, Chen, Cheng, Hu, Chen, Wang, Wenchao, Wu, Jiaxin, Hu, Zhenquan, Ye, Ling, Zou, Fengming, Liu, Feiyang, Wang, BeileiLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.6b00902
Date:
August, 2016
File:
PDF, 14.56 MB
english, 2016