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Chemically Linked Vemurafenib Inhibitors Promote an Inactive BRAFV600E Conformation
Grasso, Michael, Estrada, Michelle A., Ventocilla, Christian, Samanta, Minu, Maksimoska, Jasna, Villanueva, Jessie, Winkler, Jeffrey D., Marmorstein, RonenLanguage:
english
Journal:
ACS Chemical Biology
DOI:
10.1021/acschembio.6b00529
Date:
August, 2016
File:
PDF, 14.12 MB
english, 2016