Design, synthesis, and structure-activity relationship of novel and effective apixaban derivatives as FXa inhibitors containing 1, 2, 4-triazole/pyrrole derivatives as P2 binding element
Wang, Yong, Sun, Xiaoqing, Yang, Di, Guo, Zhuang, Fan, Xuxu, Nie, Minhua, Zhang, Feng, Liu, Yue, Li, Yue, Wang, Yulin, Gong, Ping, Liu, YajingLanguage:
english
Journal:
Bioorganic & Medicinal Chemistry
DOI:
10.1016/j.bmc.2016.09.024
Date:
September, 2016
File:
PDF, 1.65 MB
english, 2016