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Improvement of Ligand Affinity and Thermodynamic Properties by NMR-Based Evaluation of Local Dynamics and Surface Complementarity in the Receptor-Bound State
Mizukoshi, Yumiko, Takeuchi, Koh, Arutaki, Misa, Tokunaga, Yuji, Takizawa, Takeshi, Hanzawa, Hiroyuki, Shimada, IchioLanguage:
english
Journal:
Angewandte Chemie International Edition
DOI:
10.1002/anie.201607474
Date:
October, 2016
File:
PDF, 895 KB
english, 2016