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Discovery of 4-[(5-arylidene-4-oxothiazolidin-3-yl)methyl]benzoic acid derivatives active as novel potent allosteric inhibitors of protein tyrosine phosphatase 1B: In silico studies and in vitro evaluation as insulinomimetic and anti-inflammatory agents
Ottanà, Rosaria, Paoli, Paolo, Naß, Alexandra, Lori, Giulia, Cardile, Venera, Adornato, Ilenia, Rotondo, Archimede, Eleonora Graziano, Adriana Carol, Wolber, Gerhard, Maccari, RosannaLanguage:
english
Journal:
European Journal of Medicinal Chemistry
DOI:
10.1016/j.ejmech.2016.10.063
Date:
November, 2016
File:
PDF, 3.11 MB
english, 2016