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Assessment of Bromodomain Target Engagement by a Series of BI2536 Analogues with Miniaturized BET-BRET
Koblan, Luke W., Buckley, Dennis L., Ott, Christopher J., Fitzgerald, Mark E., Ember, Stuart W. J., Zhu, Jin-Yi, Liu, Shuai, Roberts, Justin M., Remillard, David, Vittori, Sarah, Zhang, Wei, SchonbrunLanguage:
english
Journal:
ChemMedChem
DOI:
10.1002/cmdc.201600502
Date:
November, 2016
File:
PDF, 845 KB
english, 2016