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Mitigation of reactive metabolite formation for a series of 3-amino-2-pyridone inhibitors of Bruton’s tyrosine kinase (BTK)
Lou, Yan, Lopez, Francisco, Jiang, Yongying, Han, Xiaochun, Brotherton, Chris, Billedeau, Roland, Gabriel, Steve, Gleason, Shelly, Goldstein, David M., Hilgenkamp, Ramona, Kocer, Buelent, Orzechowski,Volume:
27
Language:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2016.11.092
Date:
February, 2017
File:
PDF, 406 KB
english, 2017