Sulfonamides as Selective Na V 1.7 Inhibitors: Optimizing Potency and Pharmacokinetics While Mitigating Metabolic Liabilities
Weiss, Matthew M., Dineen, Thomas A., Marx, Isaac E., Altmann, Steven, Boezio, Alessandro, Bregman, Howard, Chu-Moyer, Margaret, DiMauro, Erin F., Feric Bojic, Elma, Foti, Robert S., Gao, Hua, GraceffLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.6b01851
Date:
April, 2017
File:
PDF, 987 KB
english, 2017