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Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors
Wang, Le, Pratt, John K., Soltwedel, Todd, Sheppard, George S., Fidanze, Steven D., Liu, Dachun, Hasvold, Lisa A., Mantei, Robert A., Holms, James H., McClellan, William J., Wendt, Michael D., Wada, CLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.7b00017
Date:
April, 2017
File:
PDF, 1.87 MB
english, 2017