Addressing Structural Flexibility at the A-Ring on Salvinorin A: Discovery of a Potent Kappa-Opioid Agonist with Enhanced Metabolic Stability
Sherwood, Alexander M., Crowley, Rachel Saylor, Paton, Kelly F., Biggerstaff, Andrew, Neuenswander, Benjamin, Day, Victor W., Kivell, Bronwyn M., Prisinzano, Thomas E.Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.7b00148
Date:
April, 2017
File:
PDF, 1.81 MB
english, 2017