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Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9 H -purin-9-yl)methyl)-5-methyl-3-( o -tolyl)quinazolin-4(3 H )-one (IC87114) and Its Conformationally Restricted Analogs
Lodola, Alessio, Bertolini, Serena, Biagetti, Matteo, Capacchi, Silvia, Facchinetti, Fabrizio, Gallo, Paola Maria, Pappani, Alice, Mor, Marco, Pala, Daniele, Rivara, Silvia, Visentini, Filippo, Corsi,Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.7b00247
Date:
May, 2017
File:
PDF, 2.73 MB
english, 2017