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Discovery of novel somatostatin receptor subtype 5 (SSTR5) antagonists: Pharmacological studies and design to improve pharmacokinetic profiles and human Ether-a-go-go-related gene (hERG) inhibition
Yamasaki, Takeshi, Hirose, Hideki, Yamashita, Tohru, Takakura, Nobuyuki, Morimoto, Sachie, Nakahata, Takashi, Kina, Asato, Nakano, Yoshihide, Okano Tamura, Yumiko, Sugama, Jun, Odani, Tomoyuki, ShimizLanguage:
english
Journal:
Bioorganic & Medicinal Chemistry
DOI:
10.1016/j.bmc.2017.06.003
Date:
June, 2017
File:
PDF, 1.27 MB
english, 2017