Synthesis and optimization of 4,5,6,7-tetrahydrooxazolo[4,5- c ]pyridines as potent and orally-active metabotropic glutamate receptor 5 negative allosteric modulators
Hirose, Wataru, Kato, Yoshihiro, Natsutani, Itaru, Takata, Makoto, Kitaichi, Maiko, Imai, Satoki, Hayashi, Shun, Arai, Yukiyo, Hoshino, Kohei, Yoshida, KohzoLanguage:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2017.08.030
Date:
August, 2017
File:
PDF, 644 KB
english, 2017