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Toward a generalized computational workflow for exploiting transient pockets as new targets for small molecule stabilizers: application to the homogentisate 1,2-dioxygenase mutants at the base of rare disease Alkaptonuria
Bernini, Andrea, Galderisi, Silvia, Spiga, Ottavia, Bernardini, Giulia, Niccolai, Neri, Manetti, Fabrizio, Santucci, AnnalisaLanguage:
english
Journal:
Computational Biology and Chemistry
DOI:
10.1016/j.compbiolchem.2017.08.008
Date:
August, 2017
File:
PDF, 1.95 MB
english, 2017