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Probing ligand structure-activity relationships in pregnane X receptor (PXR): efavirenz and 8-hydroxyefavirenz exhibit divergence in activation
Narayanan, Bhargavi, Lade, Julie, Heck, Carley J.S., Dietz, Kevin D., Wade, Herschel V., Bumpus, Namandje N.Language:
english
Journal:
ChemMedChem
DOI:
10.1002/cmdc.201700730
Date:
February, 2018
File:
PDF, 3.42 MB
english, 2018