Exploiting the S4-S5 specificity of human neutrophil proteinase 3 to improve the potency of peptidyl di(chlorophenyl)-phosphonate ester inhibitors: a kinetic and molecular modeling analysis
Guarino, Carla, Gruba, Natalia, Grzywa, Renata, Dyguda-Kazimierowicz, Edyta, Hamon, Yveline, Legowska, Monika, Skoreński, Marcin, Dallet-Choisy, Sandrine, Marchand-Adam, Sylvain, Kellenberger, ChristiLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.7b01416
Date:
February, 2018
File:
PDF, 1.31 MB
english, 2018