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Structure based design of a Grp94-selective inhibitor: Exploiting a key residue in Grp94 to optimize paralog-selective binding
Que, Nanette L. S., Crowley, Vincent M., Duerfeldt, Adam S, Zhao, Jinbo, Kent, Caitlin N., Blagg, Brian S.J., Gewirth, Daniel T.Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.7b01608
Date:
March, 2018
File:
PDF, 2.36 MB
english, 2018