Discovery of {4-[4,9-bis(ethyloxy)-1-oxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]-2-fluorophenyl}acetic acid (GSK726701A), a novel EP 4 receptor partial agonist for the treatment of pain
Healy, Mark P., Allan, Amanda C., Bailey, Kristin, Billinton, Andy, Chessell, Iain P., Clayton, Nicholas M., M. P. Giblin, Gerard, Kay, Melanie A., Khaznadar, Tarik, Michel, Anton D., Naylor, Alan, PrLanguage:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2018.03.091
Date:
March, 2018
File:
PDF, 770 KB
english, 2018