Discovery of N 2 -(4-Amino-cyclohexyl)-9-cyclopentyl- N 6 -(4-morpholin-4-ylmethyl-phenyl)-9 H -purine-2,6-diamine as a Potent FLT3 Kinase Inhibitor for Acute Myeloid Leukemia with FLT3 mutations
Gucky, Tomas, Řezníčková, Eva, Radosova Muchova, Tereza, Jorda, Radek, Klejova, Zuzana, Malinkova, Veronika, Berka, Karel, Bazgier, Vaclav, AJANI, HARESH, Lepsik, Martin, Divoky, Vladimir, Krystof, VlLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.7b01529
Date:
April, 2018
File:
PDF, 1.70 MB
english, 2018