BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability
Jennings, Laura E., Schiedel, Matthias, Hewings, David S., Picaud, Sarah, Laurin, Corentine M.C., Bruno, Paul A., Bluck, Joseph P., Scorah, Amy R., See, Larissa, Reynolds, Jessica K., Moroglu, MustafaVolume:
26
Language:
english
Journal:
Bioorganic & Medicinal Chemistry
DOI:
10.1016/j.bmc.2018.05.003
Date:
July, 2018
File:
PDF, 1.90 MB
english, 2018