Mechanistic kinetic modeling generates system-independent P-glycoprotein mediated transport elementary rate constants for inhibition and, in combination with 3D SIM microscopy, elucidates the importance of microvilli morphology on P-glycoprotein mediated efflux activity
Ellens, Harma, Meng, Zhou, Le Marchand, Sylvain J., Bentz, JoeLanguage:
english
Journal:
Expert Opinion on Drug Metabolism & Toxicology
DOI:
10.1080/17425255.2018.1480720
Date:
June, 2018
File:
PDF, 1.43 MB
english, 2018