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Chemical space screening around Phe 3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings
Willemse, Tom, Eiselt, Emilie, Hollanders, Karlijn, Schepens, Wim, van Vlijmen, Herman W.T., Chung, Nga N., Blais, Véronique, Holleran, Brain, Longpré, Jean-Michel, Schiller, Peter W., Maes, Bert U.W.Language:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2018.05.015
Date:
May, 2018
File:
PDF, 611 KB
english, 2018