Discovery of Potent 2-Aryl-6,7-Dihydro-5 H -Pyrrolo[1,2- a ]imidazoles as WDR5 WIN-site Inhibitors Using Fragment-Based Methods and Structure-Based Design
Wang, Feng, Jeon, Kyu Ok, Salovich, James M., Macdonald, Jonathan D, Alvarado, Joseph, Gogliotti, Rocco D., Phan, Jason, Olejniczak, Edward T, Sun, Qi, Wang, Shidong, Camper, DeMarco V., Yuh, JoannesLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.8b00375
Date:
June, 2018
File:
PDF, 6.22 MB
english, 2018