Conversion of Carbazole Carboxamide Based Reversible Inhibitors of Bruton’s Tyrosine Kinase (BTK) into Potent, Selective Irreversible Inhibitors in the Carbazole, Tetrahydrocarbazole, and a New 2,3-Dimethylindole Series
Liu, Qingjie, Batt, Douglas G., Chaudhry, Charu, Lippy, Jonathan S., Pattoli, Mark A., Surti, Neha, Xu, Songmei, Carter, Percy H., Burke, James R., Tino, Joseph A.Language:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2018.07.041
Date:
July, 2018
File:
PDF, 529 KB
english, 2018