Novel Quinazolinone Inhibitors of ALK2 Flip between Alternate Binding Modes: Structure–Activity Relationship, Structural Characterization, Kinase Profiling, and Cellular Proof of Concept
Hudson, Liam, Mui, James, Vázquez, Santiago, Carvalho, Diana M., Williams, Eleanor, Jones, Chris, Bullock, Alex N., Hoelder, SwenLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.8b00782
Date:
August, 2018
File:
PDF, 4.88 MB
english, 2018