Aiming to Miss a Moving Target: Bromo and Extra Terminal Domain (BET) Selectivity in Constrained ATAD2 Inhibitors
Bamborough, Paul, Chung, Chun-wa, Furze, Rebecca C., Grandi, Paola, Michon, Anne-Marie, Watson, Robert J., Mitchell, Darren J., Barnett, Heather, Prinjha, Rab K., Rau, Christina, Sheppard, Robert J.,Volume:
61
Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.8b00862
Date:
September, 2018
File:
PDF, 3.85 MB
english, 2018