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Discovery of N-(4-(6-acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent Fms-like Tyrosine Kinase 3 Internal Tandem Duplications (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia
Liang, Xiaofei, Wang, Beilei, Chen, Cheng, Wang, Aoli, Hu, Chen, Zou, Fengming, Yu, Kailin, Liu, Qingwang, Li, Feng, Hu, Zhenquan, Lu, Tingting, Wang, Junjie, Wang, Li, Weisberg, Ellen, Li, Lili, Xia,Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.8b01594
Date:
December, 2018
File:
PDF, 1.98 MB
english, 2018