An Activity-Based Probe Targeting Non-Catalytic, Highly Conserved Amino Acid Residues within Bromodomains
D'Ascenzio, Melissa, Pugh, Kathryn M., Konietzny, Rebecca, Berridge, Georgina, Tallant, Cynthia, Hashem, Shaima, Monteiro, Octovia, Thomas, Jason R., Schirle, Markus, Knapp, Stefan, Marsden, Brian, FeLanguage:
english
Journal:
Angewandte Chemie International Edition
DOI:
10.1002/anie.201807825
Date:
December, 2018
File:
PDF, 2.14 MB
english, 2018